Novel heterocyclic analogues of the new potent class of calcium entry blockers: 1-[[4-(aminoalkoxy)phenyl]sulfonyl]indolizines.

J, Gubin; Vogelaer H, de; H, Inion; C, Houben; J, Lucchetti; J, Mahaux; G, Rosseels; M, Peiren; M, Clinet; P, Polster

doi:10.1021/jm00062a015

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Novel heterocyclic analogues of the new potent class of calcium entry blockers: 1-[[4-(aminoalkoxy)phenyl]sulfonyl]indolizines.

Shared by NobleBlocks on May 1, 1993 • 12:00 AM UTC

Authors:

Gubin J

de Vogelaer H

Inion H

Abstract

Several heterocyclic analogues of the potent 1-[[4-(aminoalkoxy)phenyl]sulfonyl]indolizines were synthesized and evaluated for their antagonistic calcium activities in comparison with the 1-sulfonylindolizine SR 33557 and the usual calcium antagonist references verapamil, cis-(+)-diltiazem, and nife...

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